Clomiphene Citrate Overview

Main Ingredient: Clomiphene Citrate

Category: Selective Estrogen Receptor Modulator (SERM)

Formulation: Oral Tablets

Brief Summary

Originating from the triphenylethylene family, Clomiphene citrate is a renowned selective estrogen receptor modulator. This compound acts dually as both antagonist and agonist. It specifically binds and inhibits estrogen activity in most tissues, but intriguingly activates them in bone tissues, providing defense against osteoporosis.

Understanding its Function

In males, Clomiphene citrate and its counterparts function as estrogen blockers. They principally disrupt estrogen’s feedback on the hypothalamus, resulting in increased GnRH production. This domino effect spurs the pituitary gland to produce more LH and FSH hormones, leading to elevated testosterone and sperm production in the testes.

Detailedly, Clomiphene Citrate chiefly targets estrogen receptors in the pituitary gland and ovaries. It ensures that the regular estrogenic influence on pituitary function is impeded. While typical estrogens would depress FSH and LH production, Clomiphene prevents this, revitalizing the hypothalamus and pituitary gland operations swiftly.

Recommended Dosage

Post-Cycle Recovery: Commence with up to 150 mg initially, tapering to 50-25 mg over two weeks. Dosage specifics should correspond with lab results. For lighter courses, a 50 mg dose for the first week, followed by 25 mg the next week, is adequate. These recommendations should be personalized.

Boosting Testosterone Levels: Daily intake between 50 to 25 mg is recommended. Adjusting the dose based on diagnostic results is crucial. Men above 35 often find 25 mg daily effective, boosting testosterone, libido, and vitality, with minimal side effects.

Key Benefits

• Inhibits estrogen receptors, especially in the brain
• Boosts natural testosterone production
• Improves bone density
• Protects against estrogen-induced gynecomastia

Potential Adverse Effects

• Breast discomfort
• Migraines
• Stomach issues or vomiting
• Diarrhea
• Hot flashes
• Visual disturbances

Note: Side effects from Clomiphene are rare.

Product Specifications

• Persistence in Body: 5-6 days
• Consumption Frequency: Once daily

Precautionary Notes

Individuals should avoid if they:

• Have allergies to Clomiphene Citrate or its components.
• Are pregnant or breastfeeding.
• Have a history of liver disorders.
• Experience irregular vaginal bleeding, adrenal problems, non-PCOS ovarian cysts, brain tumors, or thyroid issues.

Storage Instructions

• Keep away from children.
• Store in a cool, dry place, away from sunlight.
• Maintain at room temperature.
• Use before the expiration date.